| Identifiers | ||
| Product Name | UNC0638, HMT inhibitor | |
| Catalogue No. | CM901548 | |
| Description | UNC0638 is a selective inhibitor of G9a and G9a-like protein (GLP), also known as EHMT1, with IC50's in the very low (<20) nM range. It also exhibits very weak activity against JMJD2E (IC50 ~4.5 µM), but the selectivity for G9a and GLP is over 200-fold. UNC0638 was inactive against SUV39H1, SUV39H2, EZH2), SETD7, MLL, SMYD3, DOT1L, SETD8, PRDM1, PRMT1 and PRMT3. UNC0638 exhibits only extremely weak inhibition of DNMT1 (IC50 >100 µM). | |
| CAS Number | 1255580-76-7 | |
| Formula | C30H47N5O2 | |
| MW | 509.7 Da | |
| Product Type | Inhibitor | |
| Grade | ≥98% by HPLC | |
| Storage Condition | refer to Technology Column | |
| Brand | Packing | Pricing | Quote request |
| IL | 5 mg | Inquiry | Ask Quote |
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